Tyrphostin 51, >=98%

Code: T7665-5MG D2-231

Not available outside of the UK & Ireland.

Application

Tyrphostin 51 has been used to study the inhibition of rat hepatic leptin 1.

Biochem/physiol Actions

EGFR tyrosine kinase inhibitor.<...


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Your Price
$192.51 5MG
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Not available outside of the UK & Ireland.

Application

Tyrphostin 51 has been used to study the inhibition of rat hepatic leptin 1.

Biochem/physiol Actions

EGFR tyrosine kinase inhibitor.

Tyrphostin 51 is a small molecule inhibitor of epidermal growth factor (EGF) receptor kinase function. This molecule associates with the substrate subsite of the protein tyrosine kinase (PTK) domain,.

Features and Benefits

This compound is a featured product for Kinase Phosphatase Biology research. Click here to discover more featured Kinase Phosphatase Biology products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.

Packaging

5 mg in glass bottle

25 mg in poly bottle

Preparation Note

5 mg of Tyrphostin 51 is soluble in 0.1 ml of DMSO and yields a clear, orange to red solution.

assay≥98%
biological sourcesynthetic (organic)
formpowder
Gene Informationhuman ... CDK2(1017), EGFR(1956)
InChI keyJKNOYWVMHPMBEL-UNXLUWIOSA-N
InChI1S/C13H8N4O3/c14-4-8(12(17)9(5-15)6-16)1-7-2-10(18)13(20)11(19)3-7/h1-3,18-20H,17H2/b8-1+
potency0.8 µM IC50
Quality Level200
SMILES stringNC(C(=Cc1cc(O)c(O)c(O)c1)C#N)=C(/C#N)C#N
solubilityDMSO: soluble 5 mg of Tyrphostin 51 in 0.1 ml of solvent, clear, orange to red
storage temp.2-8°C
Cas Number126433-07-6
This product has met the following criteria to qualify for the following awards:



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