Tyrphostin 51, >=98%

Code: T7665-25MG D2-231

Not available outside of the UK & Ireland.

Application

Tyrphostin 51 has been used to study the inhibition of rat hepatic leptin 1.

Biochem/physiol Actions

EGFR tyrosine kinase inhibitor.<...


 Read more

Your Price
$623.29 25MG
REQUEST

Not available outside of the UK & Ireland.

Application

Tyrphostin 51 has been used to study the inhibition of rat hepatic leptin 1.

Biochem/physiol Actions

EGFR tyrosine kinase inhibitor.

Tyrphostin 51 is a small molecule inhibitor of epidermal growth factor (EGF) receptor kinase function. This molecule associates with the substrate subsite of the protein tyrosine kinase (PTK) domain,.

Features and Benefits

This compound is a featured product for Kinase Phosphatase Biology research. Click here to discover more featured Kinase Phosphatase Biology products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.

Packaging

5 mg in glass bottle

25 mg in poly bottle

Preparation Note

5 mg of Tyrphostin 51 is soluble in 0.1 ml of DMSO and yields a clear, orange to red solution.

assay≥98%
biological sourcesynthetic (organic)
formpowder
Gene Informationhuman ... CDK2(1017), EGFR(1956)
InChI keyJKNOYWVMHPMBEL-UNXLUWIOSA-N
InChI1S/C13H8N4O3/c14-4-8(12(17)9(5-15)6-16)1-7-2-10(18)13(20)11(19)3-7/h1-3,18-20H,17H2/b8-1+
potency0.8 µM IC50
Quality Level200
SMILES stringNC(C(=Cc1cc(O)c(O)c(O)c1)C#N)=C(/C#N)C#N
solubilityDMSO: soluble 5 mg of Tyrphostin 51 in 0.1 ml of solvent, clear, orange to red
storage temp.2-8°C
Cas Number126433-07-6
This product has met the following criteria to qualify for the following awards:



PROCEED TO CHECKOUT

HAVE AN ACCOUNT? LOGIN
GUEST CHECKOUT

Proceed as a guest. You will have the option to register to access exclusive pricing and stock availability features after checkout.