(-)-N6-(2-Phenylisopropyl)adenosine, solid

Name: (-)-N6-(2-Phenylisopropyl)adenosine, solid
Brand: SIGMA-ALDRICH
SKU: P4532-50MG
Price: 298.86 USD

Code: P4532-50MG D2-231

Not available outside of the UK & Ireland.

Biochem/physiol Actions

A₁ adenosine receptor agonist. Affinity for adenosine receptor is approx. 100× that of the (+)-isomer.

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$298.86 50MG

Discontinued

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Not available outside of the UK & Ireland.
Biochem/physiol Actions
A₁ adenosine receptor agonist. Affinity for adenosine receptor is approx. 100× that of the (+)-isomer.
Features and Benefits
This compound is featured on the Adenosine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
Packaging
50, 100 mg in glass bottle
25 mg in poly bottle

color white
form solid
Gene Information human ... ADORA1(134)
InChI key RIRGCFBBHQEQQH-SSFGXONLSA-N
InChI 1S/C19H23N5O4/c1-11(7-12-5-3-2-4-6-12)23-17-14-18(21-9-20-17)24(10-22-14)19-16(27)15(26)13(8-25)28-19/h2-6,9-11,13,15-16,19,25-27H,7-8H2,1H3,(H,20,21,23)/t11-,13-,15-,16-,19-/m1/s1
potency 1.17 nM K_i for A₁ receptors (using [³H]CHA in rat forebrain preparations)
Quality Level 200
SMILES string C[C@H](Cc1ccccc1)Nc2ncnc3n(cnc23)[C@@H]4O[C@H](CO)[C@@H](O)[C@H]4O
solubility H₂O: slightly soluble 0.3 mg/mL (Solutions may be stored for several days at 4°C.), 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 1.6 mg/mL (Solutions may be stored for several days at 4°C.)
storage temp. 2-8°C

Safety Data Sheet
Safety Data Sheet for P4532-50MG
Certificate of Analysis
Sigma Certificate of Analysis

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Cas Number 38594-96-6

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(-)-N6-(2-Phenylisopropyl)adenosine, solid

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color	white
form	solid
Gene Information	human ... ADORA1(134)
InChI key	RIRGCFBBHQEQQH-SSFGXONLSA-N
InChI	1S/C19H23N5O4/c1-11(7-12-5-3-2-4-6-12)23-17-14-18(21-9-20-17)24(10-22-14)19-16(27)15(26)13(8-25)28-19/h2-6,9-11,13,15-16,19,25-27H,7-8H2,1H3,(H,20,21,23)/t11-,13-,15-,16-,19-/m1/s1
potency	1.17 nM K_i for A₁ receptors (using [³H]CHA in rat forebrain preparations)
Quality Level	200
SMILES string	C[C@H](Cc1ccccc1)Nc2ncnc3n(cnc23)[C@@H]4O[C@H](CO)[C@@H](O)[C@H]4O
solubility	H₂O: slightly soluble 0.3 mg/mL (Solutions may be stored for several days at 4°C.), 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 1.6 mg/mL (Solutions may be stored for several days at 4°C.)
storage temp.	2-8°C