Not available outside of the UK & Ireland.
Biochem/physiol Actions
CGP36742 was the first orally active GABAB-selective antagonist. The IC50 for blocking GABAergic transmission is 36 µM. Oral administration of CGP36742 in rats blocks baclofen-induced neuronal depression, and reduces learning deficit and passive avoidance in an olfactory bulbectomy depression model.
Features and Benefits
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Packaging
5, 25 mg in glass bottle
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