GR 113808, >=98% (HPLC), solid

Code: g5918-10mg D2-231

Not available outside of the UK & Ireland.

Application

GR 113808 has been used as a serotonin receptor 4 (5-HT4R) blocker to study its effects on the calcium (Ca2+) transients in rat ventricular cardiomyocy...


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Your Price
$227.51 10MG
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Not available outside of the UK & Ireland.

Application

GR 113808 has been used as a serotonin receptor 4 (5-HT4R) blocker to study its effects on the calcium (Ca2+) transients in rat ventricular cardiomyocytes. It has also been used as a 5-HT4R antagonist to study its effects on de novo enteric neurogenesis in post-embryonic zebrafish.

Biochem/physiol Actions

GR 113808 is a 5-HT4 serotonin receptor antagonist.

Features and Benefits

This compound was developed by GlaxoSmithKline. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

Legal Information

Sold for research purposes under agreement from GlaxoSmithKline

Packaging

10, 50 mg in glass bottle

assay≥98% (HPLC)
colorwhite to light pink
formsolid
Gene Informationhuman ... HTR4(3360)rat ... Htr3a(79246), Htr4(25324)
InChI keyMOZPSIXKYJUTKI-UHFFFAOYSA-N
InChI1S/C19H27N3O4S/c1-21-13-17(16-5-3-4-6-18(16)21)19(23)26-14-15-7-10-22(11-8-15)12-9-20-27(2,24)25/h3-6,13,15,20H,7-12,14H2,1-2H3
originatorGlaxoSmithKline
SMILES stringCn1cc(C(=O)OCC2CCN(CCNS(C)(=O)=O)CC2)c3ccccc13
solubilityDMSO: >20 mg/mL
storage temp.2-8°C
Cas Number144625-51-4
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