Nida-41020

Code: n8162-50mg D2-231

Not available outside of the UK & Ireland.

Biochem/physiol Actions

NIDA-41020 is a CB1 cannabinoid receptor antagonist. NIDA-41020 is structurally similar to Rimonabant, which is currently in clinical development. NID...


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Your Price
$683.17 50MG
Discontinued

Not available outside of the UK & Ireland.

Biochem/physiol Actions

NIDA-41020 is a CB1 cannabinoid receptor antagonist. NIDA-41020 is structurally similar to Rimonabant, which is currently in clinical development. NIDA-41020 is less lipophilic; developed at NIDA as a potential radioligand for CB1 receptors, Ki = 4.1 nM [in comparison AM 251, AM 281, SR 141716 (Rimonabant) have Ki of 0.6, 4.5 and 1.8 nM respectively].

assay≥97% (HPLC)
coloroff-white
formsolid
InChI keyKWDBQJRWPWTGPF-UHFFFAOYSA-N
InChI1S/C23H24Cl2N4O2/c1-15-21(23(30)27-28-12-4-3-5-13-28)26-29(20-11-8-17(24)14-19(20)25)22(15)16-6-9-18(31-2)10-7-16/h6-11,14H,3-5,12-13H2,1-2H3,(H,27,30)
Quality Level100
SMILES stringCOc1ccc(cc1)-c2c(C)c(nn2-c3ccc(Cl)cc3Cl)C(=O)NN4CCCCC4
solubilityDMSO: ~16 mg/mL, H2O: insoluble
storage temp.2-8°C
Cas Number502486-89-7
Hazard Class6.1
Un Number2811
Pack Group3
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