Non disponible en dehors du Royaume-Uni et de l'Irlande
Biochem/physiol Actions
Mixed NMDA agonist/antagonist at the polyamine site. Neuroprotective effects have been observed at high concentrations (1 mM), while neurotoxicity is observed at lower concentrations. It enhances agonist effectiveness at the strychnine-insensitive glycine site. Plays a role in cellular proliferation and differentiation; inhibits neuronal nitric oxide synthase (nNOS).
Other Notes
Polyamines: Review; Inhibitor of ATPase; DNA polymerase; ribonuclease
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