Rs-127445 Hydrochloride

Code: r2533-25mg D2-231

Not available outside of the UK & Ireland.

Biochem/physiol Actions

RS-127445 is a selective; high affinity; orally bioavailable serotonin 5-HT2B receptor antagonist. RS-127445 was found to have nanomolar affinity for ...


 Read more

Your Price
$586.74 25MG
Discontinued

Not available outside of the UK & Ireland.

Biochem/physiol Actions

RS-127445 is a selective; high affinity; orally bioavailable serotonin 5-HT2B receptor antagonist. RS-127445 was found to have nanomolar affinity for the 5-HT2B receptor (pKi=9.5) and 1,000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites.

Features and Benefits

This compound was developed by Roche. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

Packaging

5, 25 mg in glass bottle

assay≥98% (HPLC)
colorwhite to tan
formpowder
InChI keyMKJPYBJBPRFMHL-UHFFFAOYSA-N
InChI1S/C17H16FN3.ClH/c1-10(2)15-9-16(21-17(19)20-15)13-7-8-14(18)12-6-4-3-5-11(12)13;/h3-10H,1-2H3,(H2,19,20,21);1H
originatorRoche
Quality Level100
SMILES stringCl.CC(C)c1cc(nc(N)n1)-c2ccc(F)c3ccccc23
solubilityDMSO: ≥20 mg/mL
storage temp.2-8°C
Cas Number0199864-86-3
Hazard Class6.1
Un Number2811
Pack Group3
This product has met the following criteria to qualify for the following awards:



PROCEED TO CHECKOUT

HAVE AN ACCOUNT? LOGIN
GUEST CHECKOUT

Proceed as a guest. You will have the option to register to access exclusive pricing and stock availability features after checkout.